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We are analyzing https://www.nature.com/articles/s41551-017-0187-5.

Title:
Antibiotic-loaded nanoparticles targeted to the site of infection enhance antibacterial efficacy | Nature Biomedical Engineering
Description:
Bacterial resistance to antibiotics has made it necessary to resort to using antibacterial drugs that have considerable toxicities. Here, we show that conjugation of vancomycin-loaded nanoparticles with the cyclic 9-amino-acid peptide CARGGLKSC (CARG), identified via phage display on Staphylococcus aureus (S. aureus) bacteria and through in vivo screening in mice with S. aureus-induced lung infections, increases the antibacterial activity of the nanoparticles in S. aureus-infected tissues and reduces the systemic dose needed, minimizing side effects. CARG binds specifically to S. aureus bacteria but not Pseudomonas bacteria in vitro, selectively accumulates in S. aureus-infected lungs and skin of mice but not in non-infected tissue and Pseudomonas-infected tissue, and significantly enhances the accumulation of intravenously injected vancomycin-loaded porous silicon nanoparticles bearing CARG in S. aureus-infected mouse lung tissue. The targeted nanoparticles more effectively suppress staphylococcal infections in vivo relative to equivalent doses of untargeted vancomycin nanoparticles or of free vancomycin. The therapeutic delivery of antibiotic-carrying nanoparticles bearing peptides targeting infected tissues may help combat difficult-to-treat infections. Nanoparticles carrying an antibiotic and conjugated with a peptide identified via phage display that binds specifically to Staphylococcus aureus effectively suppress staphylococcal infections in vivo.
Website Age:
30 years and 10 months (reg. 1994-08-11).

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Custom-built

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🌆 Monumental Traffic: 20M - 50M visitors per month


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$531,700 per month
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Keywords {🔍}

pubmed, article, google, scholar, cas, nanoparticles, nature, aureus, central, staphylococcus, delivery, nat, access, joo, peptide, research, content, infections, med, cancer, targeted, porous, silicon, vancomycin, mater, university, information, engineering, sailor, ruoslahti, bacteria, adv, cookies, data, biomedical, infection, antibacterial, antibiotics, targeting, department, nano, usa, grant, korea, privacy, jinmyoung, teesalu, drugs, vivo, mice,

Topics {✒️}

nature portfolio journals nature portfolio permissions reprints interest policies folic-acid-based receptor targeting privacy policy advertising antibiotic-loaded nanoparticles targeted research findings included nature+ nature 527 nature scientific founder methicillin-resistant staphylococcus aureus killing multidrug-resistant bacteria iron-regulating sigma factors tumor-penetrating peptide enhances peptide-conjugated quantum dots ly6g-specific monoclonal antibody porous silicon nanoparticles tumor vasculature-targeted imaging social media business media aureus-induced lung infections author correspondence engineering program antimicrobial resistance aureus-infected tissues overcome bacterial resistance research vancomycin-loaded nanoparticles permissions vancomycin-modified nanoparticles springerlink instant access interest management based tumor-homing peptide policy asan medical center personal data tambet teesalu staphylococcus-binding peptide pseudomonas-binding peptide pseudomonas-infected tissue università di messina published maps mesoporous silicon particles porous silicon development enhance antibacterial efficiency methicillin-resistant

Questions {❓}

  • Are bloodstream leukocytes Trojan horses for the metastasis of Staphylococcus aureus?

Schema {🗺️}

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         description:Bacterial resistance to antibiotics has made it necessary to resort to using antibacterial drugs that have considerable toxicities. Here, we show that conjugation of vancomycin-loaded nanoparticles with the cyclic 9-amino-acid peptide CARGGLKSC (CARG), identified via phage display on Staphylococcus aureus (S. aureus) bacteria and through in vivo screening in mice with S. aureus-induced lung infections, increases the antibacterial activity of the nanoparticles in S. aureus-infected tissues and reduces the systemic dose needed, minimizing side effects. CARG binds specifically to S. aureus bacteria but not Pseudomonas bacteria in vitro, selectively accumulates in S. aureus-infected lungs and skin of mice but not in non-infected tissue and Pseudomonas-infected tissue, and significantly enhances the accumulation of intravenously injected vancomycin-loaded porous silicon nanoparticles bearing CARG in S. aureus-infected mouse lung tissue. The targeted nanoparticles more effectively suppress staphylococcal infections in vivo relative to equivalent doses of untargeted vancomycin nanoparticles or of free vancomycin. The therapeutic delivery of antibiotic-carrying nanoparticles bearing peptides targeting infected tissues may help combat difficult-to-treat infections. Nanoparticles carrying an antibiotic and conjugated with a peptide identified via phage display that binds specifically to Staphylococcus aureus effectively suppress staphylococcal infections in vivo.
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      headline:Antibiotic-loaded nanoparticles targeted to the site of infection enhance antibacterial efficacy
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